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抑制剂 & 化合物

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天然产物

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Cat. No. Product Name Target Signaling Pathways
T63901 Axl-IN-8

Axl-IN-8 (NO.1) 是 AXL 的有效抑制剂 (IC50<1 nM),也能够抑制 c-MET (IC50: 1-10 nM)。Axl-IN-8 能够抗 BaF3/TEL-AXL 细胞 (IC50<10 nM)、MKN45 细胞 (IC50: 226.6 nM) 和 EBC-1 细胞 (IC50: 120.3 nM) 的增殖。

化合物

Axl-IN-8
Cat.No: T63901
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T36886 Pestalotin

Pestalotin is a fungal metabolite originally isolated from P. cryptomeriaecola with diverse biological activities. It induces reducing sugar release in embryoless rice endosperms when used at concentrations ranging from 3 to 100 mg/L and enhances growth of rice seedlings (O. sativa) when used in combination with gibberellin A3 at concentrations ranging from 30 to 500 mg/L. Pestalotin has antifungal activity, reducing the growth of C. albicans, C. neoformans, T. rubrum, and A. fumigatus (MICs = 1...

天然产物

Pestalotin
Cat.No: T36886
Synonym:
Target:
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