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5

抑制剂 & 化合物

2

天然产物

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重组蛋白

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Cat. No. Product Name Target Signaling Pathways
T76931 Birtamimab

Birtamimab (NEOD001) 为一研究性单克隆抗体,特异性且选择性地靶向并清除淀粉样蛋白,主要应用于轻链淀粉样变性的研究。
T83106 Anselamimab

Anselamimab (CAEL-101) 为一种靶向血清淀粉样蛋白 A1 (SAA1) 的人源 IgG1-κ 抗淀粉样蛋白原纤维抗体。
T63389 AHR antagonist 5 hemimaleate

AHR antagonist 5 hemimaleate 是一种口服具有活力的芳香烃受体 (AHR) 的有效拮抗剂 (IC50< 0.5 μM)。AHR antagonist 5 hemimaleate 联合检测点抑制剂 anti-PD-1 对肿瘤生长表现出抑制作用。
T75656 Calcimycin hemimagnesium

Calcimycin (A-23187) hemimagnesium,一种具有抗生素功能的独特二价阳离子离子载体(例如钙离子和镁离子),通过提高细胞内钙浓度而诱导Ca2+依赖性细胞死亡。该化合物还能抑制革兰氏阳性细菌和部分真菌生长,同时抑制ATP酶活性并解耦哺乳动物细胞的氧化磷酸化(OXPHOS),触发细胞凋亡(apoptosis)。
T37279 1-Methyl-4-imidazoleacetic Acid (hydrochloride)

1-Methyl-4-imidazoleacetic acid (MIMA) is a stable metabolite of histamine that is produced by the oxidation of the primary metabolite, N-methylhistamine. Urinary levels of MIMA are commonly measured to evaluate histamine secretion, particularly in the context of systemic mastocytosis.

化合物

Birtamimab
Cat.No: T76931
Synonym:
Target:
Anselamimab
Cat.No: T83106
Synonym:
Target:
AHR antagonist 5 hemimaleate
Cat.No: T63389
Synonym:
Target:
Calcimycin hemimagnesium
Cat.No: T75656
Synonym:
Target:
1-Methyl-4-imidazoleacetic Acid (hydrochloride)
Cat.No: T37279
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T19281L Dihydroxyacetone phosphate hemimagnesium salt hydrate

Dihydroxyacetone phosphate hemimagnesium salt hydrate(57-04-5 free base)

Others Others
Dihydroxyacetone phosphate hemimagnesium salt hydrate 也称为磷酸二羟基丙酮或 3-羟基-2-氧代丙基磷酸。 Dihydroxyacetone phosphate hemimagnesium salt hydrate 存在于从细菌到人类的所有生物中。在人类体内, Dihydroxyacetone phosphate hemimagnesium salt hydrate参与许多酶促反应。 Dihydroxyacetone phosphate hemimagnesium salt hydrate 已被研究用于治疗淋巴瘤、大细胞淋巴瘤、弥漫性淋巴瘤。
T73763 Dihydroxyacetone phosphate hemimagnesium hydrate

Dihydroxyacetone phosphate 是脂质生物合成和糖酵解中的重要中间产物,参与卡尔文循环和糖酵解等多种代谢途径。此化合物与醛缩酶缺乏症,一种先天性代谢缺陷,相关。

天然产物

Dihydroxyacetone phosphate hemimagnesium salt hydrate
Cat.No: T19281L
Synonym: Dihydroxyacetone phosphate hemimagnesium salt hydrate(57-04-5 free base)
Target: Others
Dihydroxyacetone phosphate hemimagnesium hydrate
Cat.No: T73763
Synonym:
Target:
Cat. No. Product Name Species Expression System
TMPY-02384 MTSS1 Protein, Human, Recombinant (aa1-250, His & MBP)

metastasis suppressor 1,MIMB,MIM,MIMA

Human E. coli
MTSS1 (Metastasis suppressor 1), also known as Missing in metastasis (MIM), is a tissue-specific regulator of plasma membrane dynamics. MTSS1 is well described for its function as a metastasis suppressor gene and is expressed in a variety of tissues. MTSS1 might be involved in shaping neuronal membranes in vivo. MTSS1 deforms phosphoinositide-rich membranes through its I-BAR domain and interacts with actin monomers through its WH2 domain. MTSS1/MIM was first identified as a metastasis suppressor...

重组蛋白

MTSS1 Protein, Human, Recombinant (aa1-250, His & MBP)
Cat.No: TMPY-02384
Species: Human
Expression System: E. coli
TargetMol Loading
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