Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T18308 |
MC-Gly-Gly-Phe
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MC-Gly-Gly-Phe 是一种用于抗体-药物偶联物的可切割接头。 | |||
T8667 |
MC-Gly-Gly-Phe-Gly
DSN28369 |
Others | Others |
MC-Gly-Gly-Phe-Gly (DSN28369) 是一种可降解的 ADC linker,是一种异双功能接头,可用于制备抗体药物偶联物。 | |||
T40257 |
Mc-Gly-Gly-Phe-Gly-PAB-OH
Mc-GGFG-PAB-OH,Mc-Gly-Gly-Phe-Gly-PAB-OH |
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Mc-Gly-Gly-Phe-Gly-PAB-OH, also known as Mc-GGFG-PAB-OH, serves as a cleavable ADC linker exclusively employed in the synthesis of antibody-drug conjugates (ADCs). | |||
T39064 |
MC-Gly-Gly-Phe-Gly-NH-CH2-O-CH2COOH
MC-Gly-Gly-Phe-Gly-NH-CH2-O-CH2COOH |
Others | Others |
MC-Gly-Gly-Phe-Gly-NH-CH2-O-CH2COOH is an ADC linker commonly employed in ADC synthesis. This cleavable linker plays a fundamental role in the conjugation process of antibody-drug conjugates (ADCs). | |||
T77833 |
Mc-Gly-Gly-Phe-Gly-PAB-OH TFA
Mc-GGFG-PAB-OH TFA |
Others | Others |
Mc-Gly-Gly-Phe-Gly-PAB-OH (Mc-GGFG-PAB-OH) TFA为可降解的ADC linker,适用于抗体偶联活性分子(ADC)的合成。 | |||
T77858 |
MC-Gly-Gly-Phe-Gly-Cyclobutanecarboxylic-Exatecan
|
Others | Others |
MC-Gly-Gly-Phe-Gly-Cyclobutanecarboxylic-Exatecan是一个构成抗体药物偶联物(ADC)活性部分的化合物,由ADC连接子(MC-Gly-Gly-Phe-Gly-Cyclobutanecarboxylic)与DNA拓扑异构酶I抑制剂Exatecan通过化学键合形成。此合成ADC主要应用于癌症研究领域。 | |||
T74723 |
MC-Gly-Gly-Phe-Gly-(R)-Cyclopropane-Exatecan
|
Others | Others |
MC-Gly-Gly-Phe-Gly-(R)-Cyclopropane-Exatecan 是一种抗体偶联活性分子的一部分 (drug-linker conjugate for ADC),包含 Exatecan 。Exatecan 是一种 DNA 拓扑异构酶 I (Topoisomerase I) 抑制剂 (IC50=2.2 μM)。 | |||
T74724 |
MC-Gly-Gly-Phe-Gly-(S)-Cyclopropane-Exatecan
|
Others | Others |
MC-Gly-Gly-Phe-Gly-(R)-Cyclopropane-Exatecan 是抗体偶联活性分子的一部分 (drug-linker conjugate for ADC),包含 Exatecan 。Exatecan 是一种 DNA 拓扑异构酶 I (Topoisomerase I) 抑制剂 (IC50=2.2 μM)。 | |||
T77879 |
MC-Gly-Gly-Phe-Gly-amide-cyclopropanol-amide-Exatecan
|
Others | Others |
MC-Gly-Gly-Phe-Gly-amide-cyclopropanol-amide-Exatecan 是一种抗体活性分子偶联物。 |