Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T27985 |
MC-70
MC70,MC 70 |
||
MC-70 is a potent P-glycoprotein (P-gp) inhibitor (EC50 = 0.69 μM). | |||
T69897 |
MC-70 hydrochloride
|
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MC-70 hydrochloride is a potent P-gp inhibitor with good selectivity towards BCRP pump (EC50 values 0.05 μM, 0.69 μM, 9.3 μM, and 73 μM for Caco-2, MDR1, MRP1, and BCRP inhibition, respectively). | |||
T69896 |
Sabarubicin
MEN 10755 |
||
Sabarubicin 是一种阿霉素双糖类似物,具有显著的抗肿瘤活性。Sabarubicin 作为一种拓扑异构酶 II 毒药比阿霉素更有效,并在较低的细胞内浓度下刺激 DNA 片段。 |