Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T78094 |
Eglumegad hydrochloride
LY354740 hydrochloride,Eglumetad hydrochloride |
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Eglumegad (LY354740) hydrochloride是一种高效且选择性的group II (mGlu2/3) receptor激动剂,其对人mGlu2和mGlu3受体的IC50值分别是5和24 nM。该化合物能够保护神经元不受NMDA毒性影响,并表现出抗焦虑及抗精神病样作用。 |