Cat. No. | Product Name | Target | Signaling Pathways |
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TP1139 |
Orexin B, human
Human orexin B |
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Orexin B, human is an endogenous agonist at Orexin receptor with Kis of 420 and 36 nM for OX1 and OX2, respectively. Orexin B is a hypothalamatic neuropeptide stimulating food intake in rats. | |||
TP1138 |
Orexin B, human TFA (205640-91-1 free base)
Orexin B, human TFA,Human orexin B TFA |
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Orexin B, human (TFA) is an endogenous agonist at Orexin receptor with Kis of 420 and 36 nM for OX1 and OX2. | |||
TP1975 |
[Ala11,D-Leu15]-Orexin B(human)
[Ala11,D-Leu15]-Orexin B |
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Highly potent and selective OX2 receptor agonist; displays 400-fold selectivity over OX1 receptors. EC50 values are 0.13 and 52 nM for human OX2 and OX1 receptors respectively. | |||
T75920 |
Orexin B, human TFA
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Orexin B, human (TFA) 是 Orexin 受体的内源性激动剂,与 OX1和 OX2结合的 Ki 值分别为 420 和 36 nM。 | |||
T75921 |
[Ala11,D-Leu15]-Orexin B(human) TFA
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[Ala11,D-Leu15]-Orexin B(human) TFA为高效的orexin-2 receptor (OX2)选择性激动剂。其对OX2展现出比OX1 (52 nM) 高达400倍的较高选择性(EC50=0.13 nM)。 |