Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
TP1138 |
Orexin B, human TFA (205640-91-1 free base)
Orexin B, human TFA,Human orexin B TFA |
||
Orexin B, human (TFA) is an endogenous agonist at Orexin receptor with Kis of 420 and 36 nM for OX1 and OX2. | |||
T75920 |
Orexin B, human TFA
|
||
Orexin B, human (TFA) 是 Orexin 受体的内源性激动剂,与 OX1和 OX2结合的 Ki 值分别为 420 和 36 nM。 | |||
T75921 |
[Ala11,D-Leu15]-Orexin B(human) TFA
|
||
[Ala11,D-Leu15]-Orexin B(human) TFA为高效的orexin-2 receptor (OX2)选择性激动剂。其对OX2展现出比OX1 (52 nM) 高达400倍的较高选择性(EC50=0.13 nM)。 |