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Cat. No. | Product Name | Target | Signaling Pathways |
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T62267 |
18-Deoxyherboxidiene
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18-Deoxyherboxidiene (RQN-18690A) 是一种有效的血管生成抑制剂。18-Deoxyherboxidiene 能够选择性作用于 SF3b,其中 SF3b 是剪接体中 U2 小核核糖核蛋白 (snRNP) 的亚复合体。18-Deoxyherboxidiene 对人脐静脉内皮细胞 (HUVEC) 的迁移和管形成具有抑制作用,且无明显的细胞毒性。18-Deoxyherboxidiene 具有潜力进行癌症的研究。 |
Cat. No. | Product Name | Target | Signaling Pathways |
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T36749 |
Herboxidiene
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Herboxidiene is a polyketide originally isolated from S. chromofuscus that has diverse biological activities.[1],[2,][3],[4],[5] It inhibits growth of HeLa S3, SK-MEL-2, PC3, A549, and EBC-1 cells with GI50 values ranging from 7.4 to 62 nM.3 Herboxidiene is cytostatic against human umbilical vein endothelial cells (HUVECs; (IC50 = 26 nM)) and inhibits VEGF-induced invasion and tube formation of serum-starved HUVECs in a concentration-dependent manner, indicating antiangiogenic activity.[4] Herbo... |