Cat. No. | Product Name | Target | Signaling Pathways |
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TP2015 |
HS014
HS 014 |
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Potent and selective melanocortin MC4 receptor antagonist (Ki values are 3.16, 108, 54.4 and 694 nM for cloned human MC4, MC1, MC3 and MC5 receptors respectively). Increases food intake in rats and nociception in mice following central administration in v | |||
T75853 |
HS014 TFA
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HS014 TFA 是一种高效、选择性的黑素皮质素-4(MC4)受体拮抗剂,对人 MC4、MC1、MC3 和 MC5 受体的Ki 值分别为 3.16、108、54.4 和 694 nM。HS014 TFA 增加自由喂养大鼠的食物摄取量。 |