Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T2260 |
GW9662
2-氯-5-硝基-N-苯基苯酰胺,TIMTEC-BB SBB006523,GW 9662 |
PPAR | DNA Damage/DNA Repair; Metabolism |
GW9662 (TIMTEC-BB SBB006523) 是一种特异性 PPARγ 拮抗剂,IC50值为3.3 nM,在细胞中对 PPARγ 的功能选择性是 PPARα/δ 的 10 到 1000 倍。 | |||
T24827 |
SR 16832
SR-16832,SR16832 |
PPAR | DNA Damage/DNA Repair; Metabolism |
SR 16832 是一种化学合成中的砌块 | |||
T35468 |
(±)19(20)-EDP Ethanolamide
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(±)19(20)-EDP ethanolamide is an ω-3 endocannabinoid epoxide and cannabinoid (CB) receptor agonist (EC50s = 108 and 280 nM for CB1 and CB2, respectively). It is produced through direct epoxygenation of docosahexaenoyl ethanolamide by cytochrome P450 (CYP) epoxygenases. (±)19(20)-EDP ethanolamide (25 μM) reduces the viability of 143B metastatic osteosarcoma cells. It decreases the production of IL-6 and increases the production of IL-10 when used at concentrations ranging from 2.5 to 10 μM in BV-... |