Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T8861 |
GSK199
|
PAD | Chromatin/Epigenetic |
GSK199 是可逆的 PAD4选择性抑制剂,当缺少钙离子时,其 IC50值为 200 nM。 | |||
T71343 |
GSK1997132B
|
||
GSK1997132B is a potent, metabolically stable and centrally penetrant PPARγ partial agonist. |