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Cat. No. Product Name Target Signaling Pathways
T32005 GSK1842799

GSK 1842799

GSK1842799 is a selective S1P1 receptor agonist with good oral bioavailability.
T71069 GSK1842799 HCl

GSK1842799 is a selective S1P1 receptor agonist for multiple sclerosis. Upon phosphorylation, GSK1842799 showed subnanomole S1P1 agonist activity with >1000× selectivity over S1P3. GSK1842799 demonstrated good oral bioavailability. On the basis of the favorable in vitro ADME and in vivo PK/PD properties as well as broad toxicology evaluations, GSK1842799 was selected as a candidate for further clinical.
T71067 MK-1775 hemihydrate

MK-1775 hemihydrate is a WEE1 inhibitor with potential antineoplastic sensitizing activity.

化合物

GSK1842799
Cat.No: T32005
Synonym: GSK 1842799
Target:
GSK1842799 HCl
Cat.No: T71069
Synonym:
Target:
MK-1775 hemihydrate
Cat.No: T71067
Synonym:
Target:
TargetMol Loading
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