Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T73854 | GB-110 hydrochloride | ||
GB-110 hydrochloride 是一种有效的,具有口服活性的,非肽类的 protease activated receptor2 (PAR2)激动剂。GB-110 hydrochloride 选择性诱导 PAR2介导的 HT29 细胞内 Ca2+释放,EC50值为 0.28 μM。 | |||
T11369L |
GB-110 hydrochloride (1252806-70-4 free base)
GB-110 hydrochloride |
Others | Others |
GB-110 hydrochloride selectively induces PAR2-mediated intracellular Ca2+ release in HT29 cells with an EC50 of 0.28 μM. GB-110 hydrochloride is a potent, orally active, and nonpeptidic protease activated receptor 2 (PAR2) agonist. |