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抑制剂 & 化合物

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天然产物

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Cat. No. Product Name Target Signaling Pathways
T37791 A-971432

A-971432 is a sphingosine-1-phosphate receptor 5 (S1P5) agonist that is selective for S1P5 over S1P1 and S1P3 (IC50s = 0.006, 0.362, and >10 &#181M, respectively). It inhibits forskolin-induced cAMP production in CHO cells expressing S1P5 (EC50 = 4.1 nM). A-971432 (1 &#181M) increases electrical resistance of hCMEC/D3 cells in an in vitro blood-brain barrier model, indicating enhanced barrier integrity, and attenuates blood-brain barrier leakage in an R6/2 transgenic mouse model of Huntington’s ...

化合物

A-971432
Cat.No: T37791
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
TN4074 Forskolin J

Others Others
Forskolin J 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN4074,CAS号为 81873-08-7。

天然产物

Forskolin J
Cat.No: TN4074
Synonym:
Target: Others
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