Cat. No. | Product Name | Target | Signaling Pathways |
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T24067 |
Flt3 Inhibitor IV
Flt3 Inhibitor-IV,Flt3-IN-IV |
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Flt3 Inhibitor IV is a potent ATP-competitive Flt3 inhibitor. | |||
T29062 |
UNC3133
UNC 3133,UNC-3133 |
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UNC3133 is a potent and selective Mer tyrosine kinase (MerTK) inhibitor with IC50 Mer 3.0 nM; Axl 17nM; Tyro 3.31 nM; FLT3 6.6 nM; PO Cmax = 0.023; IV T1/2 = 1.59 h, %F = 16. Mer tyrosine kinase (MerTK) is aberrantly elevated in various tumor cells and ha |