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Cat. No. Product Name Target Signaling Pathways
T11221 ERAP1-IN-1

Others Others
ERAP1-in-1 是一种内质网氨基肽酶 1 (ERAP1) 抑制剂,能竞争性地抑制 ERAP1 对代表性生物底物九聚物肽的作用。
T27160 DG026

DG 026,DG-026

DG026 is a IRAP inhibitor. DG026 ables to selectively downregulate IRAP-dependent cross-presentation by dendritic cells but leave ERAP1-dependent cross-presentation unaffected.
T69998 DG046

DG046 is a novel potent phosphinic pseudopeptide ERAP1 inhibitor, binding in the ERAP1 active site, being stabilized by an unusual extensive network of π-stacking interactions
T63546 DG013A

DG013A 是次膦酸三肽模拟抑制剂,能够作用于 ERAP1 (IC50: 33 nM) 和 ERAP2 (IC50: 11 nM)。DG013A 能够用研究自身免疫性疾病和癌症。

化合物

ERAP1-IN-1
Cat.No: T11221
Synonym:
Target: Others
DG026
Cat.No: T27160
Synonym: DG 026,DG-026
Target:
DG046
Cat.No: T69998
Synonym:
Target:
DG013A
Cat.No: T63546
Synonym:
Target:
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