Cat. No. | Product Name | Target | Signaling Pathways |
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T69907 |
EML-405
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EML-405 is a small-molecule inhibitor of SPIN1 ( Kd of 14 uM). | |||
T69906 |
PEAQX sodium
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PEAQX, also known as NVP-AAM077; is a competitive antagonist at the NMDA receptor. Although originally described as 100-fold selective for GluN1/GluN2A receptors vs. GluN1/GluN2B receptors, more detailed studies of the Ki of PEAQX revealed it only shows a 5 fold difference in affinity for GluN1/GluN2A vs. GluN1/GluN2B receptors. It is also a potent anticonvulsant in animal tests. |