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Cat. No. Product Name Target Signaling Pathways
T61732 EGFR/HER2-IN-6

EGFR/HER2-IN-6 (compound 43) is a dual EGFR/HER2 and DHFR inhibitor with potent activity against EGFR kinase, HER2 kinase, and DHFR, characterized by IC50 values of 0.122 μM, 0.078 μM, and 0.585 μM, respectively. This compound displays notable anticancer properties in various cancer cell lines, while demonstrating a favorable safety profile and selectivity indices. Consequently, EGFR/HER2-IN-6 holds promise as a valuable tool in cancer research [1].
T63441 HER2-IN-6

HER2-IN-6HER2 的有效抑制剂。HER2-IN-6 具有潜力进行野生和/或突变 EGFR 和/或 HER2 激酶介导的肿瘤的研究。

化合物

EGFR/HER2-IN-6
Cat.No: T61732
Synonym:
Target:
HER2-IN-6
Cat.No: T63441
Synonym:
Target:
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