购物车

搜索结果

Search Results for " distamycin a "

2

抑制剂 & 化合物

1

天然产物

如果没找到您满意的产品或者您对产品有其他要求,可以联系我们专业顾问为您提供针对性的合理建议。     QQ咨询       网站留言咨询

提交您的定制咨询

点击图片重新获取验证码
Cat. No. Product Name Target Signaling Pathways
T68151 Tallimustine

FCE 24517

Tallimustine (FCE 24517),一种 distamycin-A 衍生物,是一种抗癌剂。
T69978 Brostallicin HCl

Brostallicin is a synthetic, alpha-bromoacrylic, second-generation minor groove binder (MGB), related to distamycin A, with potential antineoplastic activity. Brostallicin binds to DNA minor groove DNA, after having formed a highly reactive glutathione (GSH)-brostallicin complex in the presence of the enzyme glutathione S-transferase (GST), which is overexpressed in cancer cells; DNA replication and cell division are inhibited, resulting in tumor cell death. Compared to typical MGBs, this agent ...

化合物

Tallimustine
Cat.No: T68151
Synonym: FCE 24517
Target:
Brostallicin HCl
Cat.No: T69978
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T73730 Distamycin A

Distamycin A (NSC-82150)为一种寡肽抗生素及小沟结合剂,其结合B型DNA,并倾向于A/T富集区。Distamycin A能调节烯二炔诱导DNA切割位点并促进细胞凋亡。

天然产物

Distamycin A
Cat.No: T73730
Synonym:
Target:
TargetMol Loading
联系我们
400-820-0310

上海市静安区江场三路238号8楼