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Cat. No. Product Name Target Signaling Pathways
T18601 Desmethyl-QCA276

PROTAC BRD4-binding moiety 4

Others Others
Desmethyl-QCA276, the QCA276-based moiety, binds to cereblon ligand via a linker to form PROTAC to degrade BET. QCA276 is a BET inhibitor with an IC50 of 10 nM, and with a Ki of 2.3 nM[1].

化合物

Desmethyl-QCA276
Cat.No: T18601
Synonym: PROTAC BRD4-binding moiety 4
Target: Others
TargetMol Loading
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