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Cat. No. Product Name Target Signaling Pathways
T62068 Chitin synthase inhibitor 1

Chitin synthase inhibitor 1 是有效的、选择性的几丁质合酶 (CHS) 抑制剂,IC50值为0.12 mM。Chitin synthase inhibitor 1 强效抑制耐药真菌变体。
T61188 Chitin synthase inhibitor 2

Chitin synthase inhibitor 2 (compound 2b) is a highly potent inhibitor of chitin synthase, with an IC50 value of 0.09 mM and a K i value of 0.12 mM. This compound exhibits antimicrobial activities in vitro and demonstrates synergistic or additive effects when combined with fluconazole or polyoxin B [1].
T78886 Chitin synthase inhibitor 14

Chitin synthase inhibitor 14 (compound 4n),一种CHS抑制剂,展现出优异的抗真菌活性和对耐药真菌变异的有效抗性。
T61398 Chitin synthase inhibitor 3

Chitin synthase inhibitor 3 (compound 2d) 是一种高效的chitin synthase抑制剂,具有0.16 mM的IC50值,并对candida albicans显示出1 μg/mL的MIC,表现出抗真菌活性。
T79481 Chitin synthase inhibitor 13

Chitin synthase inhibitor 13 (compound 12g) 为非竞争性几丁质合酶抑制剂,其IC50为106.7 μM,展现出广谱抗真菌活性。
T74956 Chitin synthase inhibitor 10

Chitin synthase inhibitor 10为一种高效的几丁质合酶(CHS)抑制剂,具有0.11 mM的IC50,表现出显著的CHS抑制活性。作为抗真菌剂,该化合物对包括C. albicans和C. neoformans在内的耐药真菌变体有效,适合用于侵袭性真菌感染(IFI)研究。

化合物

Chitin synthase inhibitor 1
Cat.No: T62068
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Target:
Chitin synthase inhibitor 2
Cat.No: T61188
Synonym:
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Chitin synthase inhibitor 14
Cat.No: T78886
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Chitin synthase inhibitor 3
Cat.No: T61398
Synonym:
Target:
Chitin synthase inhibitor 13
Cat.No: T79481
Synonym:
Target:
Chitin synthase inhibitor 10
Cat.No: T74956
Synonym:
Target:
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