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Cat. No. Product Name Target Signaling Pathways
T35479 CRBN-6-5-5-VHL

PROTACs PROTAC
Potent and selective cereblon degrader (DC50 = 1.5 nM). Induces complete degradation of cereblon in MM1S cells. Comprises a cereblon E3 ligase ligand joined by a linker to a ligand for the E3 ligase VHL. Cell-permeable. Steinebach et al (2019) PROTAC-mediated crosstalk between E3 ligases. Chem.Commun.(Camb) 55 1821 PMID:30672516

化合物

CRBN-6-5-5-VHL
Cat.No: T35479
Synonym:
Target: PROTACs
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