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Cat. No. Product Name Target Signaling Pathways
T21584 CP 465022

iGluR Membrane transporter/Ion channel; Neuroscience
CP 465022 hydrochloride 是强效的、选择性的AMPA 受体非竞争性拮抗剂,具有抗惊厥活性。CP 465022 hydrochloride 在大鼠皮层神经元中抑制Kainate 诱导的反应 (IC50= 25 nM)。
T21875 CP-465022 (maleate)

CP-465022 Maleate is a potent, selective, noncompetitive AMPA receptor antagonist with anticonvulsant activity. It effectively counters the Kainate-induced response in rat cortical neurons, exhibiting an IC 50 of 25 nM. As such, CP-465022 Maleate presents a valuable instrument for studying the involvement of AMPA receptors in various physiological and pathophysiological processes [1] [2].

化合物

CP 465022
Cat.No: T21584
Synonym:
Target: iGluR
CP-465022 (maleate)
Cat.No: T21875
Synonym:
Target:
TargetMol Loading
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