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6

抑制剂 & 化合物

1

重组蛋白

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Cat. No. Product Name Target Signaling Pathways
T63520 ChemR23-IN-2

ChemR23-IN-2 是强效的、口服具有活力的 ChemR23 抑制剂 (IC50: 3.2 nM)。
T63195 ChemR23-IN-4

ChemR23-IN-4 是口服具有活力的ChemR23的有效抑制剂,能够作用于人 ChemR23 (IC50: 17 nM)。
T63347 ChemR23-IN-1

ChemR23-IN-1 是 ChemR23 抑制剂,能够作用于人和小鼠 ChemR23,他们的IC50值分别为 38 nM 和 100 nM。ChemR23-IN-1 能够阻碍体外 Chemerin 触发的 CAL-1 趋化性。
T72933 ChemR23-IN-3

ChemR23-IN-3 是一种有效的基于噻唑的ChemR23抑制剂,其IC80值为 12 nM。
TP1617L Chemerin-9 (149-157) acetate

Chemerin-9 (149-157) acetate (676367-27-4 free base)

Others Others
Chemerin-9 (149-157) acetate (676367-27-4 free base) 对应于加工的 chemerin 的 C 末端,保留了全尺寸蛋白质的大部分活性和关于对 chemerinR 的激动。它是 ChemR23 (chemerinR) 的天然配体。
TP1617 Chemerin-9 (149-157)

Chemerin-9 149-157

The nonapeptide 149,YFPGQFAFS157 (chemerin-9), corresponding to the C terminus of processed chemerin, retained most of the activity of the full-size protein, with regard to agonism toward the chemerinR.the natural ligand of ChemR23 (chemerinR).

化合物

ChemR23-IN-2
Cat.No: T63520
Synonym:
Target:
ChemR23-IN-4
Cat.No: T63195
Synonym:
Target:
ChemR23-IN-1
Cat.No: T63347
Synonym:
Target:
ChemR23-IN-3
Cat.No: T72933
Synonym:
Target:
Chemerin-9 (149-157) acetate
Cat.No: TP1617L
Synonym: Chemerin-9 (149-157) acetate (676367-27-4 free base)
Target: Others
Chemerin-9 (149-157)
Cat.No: TP1617
Synonym: Chemerin-9 149-157
Target:
Cat. No. Product Name Species Expression System
TMPH-01082 CMKLR1 Protein, Human, Recombinant (His)

CMKLR1,G-protein coupled receptor ChemR23,...

Human E. coli
CMKLR1 Protein, Human, Recombinant (His) is expressed in E. coli expression system with N-10xHis tag. The predicted molecular weight is 45.1 kDa and the accession number is Q99788.

重组蛋白

CMKLR1 Protein, Human, Recombinant (His)
Cat.No: TMPH-01082
Species: Human
Expression System: E. coli
TargetMol Loading
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