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抑制剂 & 化合物

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Cat. No.	Product Name	Target	Signaling Pathways
T25242	Chlornaphazine CB 1048,CB-1048,R 48,Erysan,CB1048
	Chlornaphazine is an antineoplastic and has been identified as a human carcinogen.
T72011	CB-892
	CB-892 is a novel inhibitor of hiv-1 gene expression
T61402	PGN36
	PGN36 (Compound 18) is a potent and highly selective antagonist of the cannabinoid CB 2 receptor (CB 2 R). It exhibits exceptional affinity for CB 2 R, with a Ki value of 0.09 μM [1].
T38028	(R)-(+)-Docosahexaenyl-1'-Hydroxy-2'-Propylamide
	N-Acyl ethanolamines (NAEs) have diverse biological actions that are strongly affected by the associated acyl group. Docosahexaenoyl ethanolamide (DHEA) has potential signaling roles in cancer, inflammation, and neurological development and functioning. At least some of DHEA's effects are mediated through cannabinoid (CB) receptors, while some NAEs also act as vanilloid receptor agonists and voltage-gated K+ channel blockers. (R)-(+)-Docosahexaenyl-1'-hydroxy-2'-propylamide is a homolog of DHEA,...
T32337	JWH-167 JWH 167,JWH167
	JWH 167, a synthetic cannabinoid (CB), has moderate affinities for central CB1 (Ki = 90 nM) and peripheral CB2 (Ki = 159 nM) receptors. Its physiological and toxicological properties have not been evaluated. This product is only applied for forensic and r
T38030	(R)-AM1241 (R)-AM1241
	(R)-AM1241 binds to cannabinoid (CB) receptors and has greater than 100-fold selectivity for the CB2 over the CB1 receptor (Kis = 15 and 5,000 nM, respectively, in a membrane assay using human receptors). (R)-AM1241 acts as an agonist at human CB2 receptors (EC50 = 118 nM) but an inverse agonist at rat and mouse CB2 receptors (EC50s = 315 and 341 nM, respectively). Similar to the racemate AM1241 , (R)-AM1241 produces antinociception to thermal, but not mechanical, pain in rats. The pain-reducing...

化合物

Chlornaphazine

Cat.No: T25242

Synonym: CB 1048,CB-1048,R 48,Erysan,CB1048

(R)-(+)-Docosahexaenyl-1'-Hydroxy-2'-Propylamide

Synonym: JWH 167,JWH167

Target:

(R)-AM1241

Cat.No: T38030

Synonym: (R)-AM1241

Target:

Species：

Expression System：

Tag：

Cat. No.	Product Name	Species	Expression System
TMPH-03256	CNR1 Protein, Rat, Recombinant (His) Skr6,Brain-type cannabinoid recep...	Rat	E. coli
	CNR1 Protein, Rat, Recombinant (His) is expressed in E. coli expression system with N-10xHis tag. The predicted molecular weight is 58.9 kDa and the accession number is P20272.
TMPH-01035	CNR1 Protein-VLP, Human, Recombinant (His) Cnr1,Skr6,CB1,CB-R	Human	HEK293 Cells
	CNR1 Protein-VLP, Human, Recombinant (His) is expressed in HEK293 mammalian cells with C-10xHis tag. The predicted molecular weight is 54.6 kDa and the accession number is P21554.