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4

抑制剂 & 化合物

1

天然产物

1

重组蛋白

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Cat. No. Product Name Target Signaling Pathways
T125203 Excavatin M

T70066 Pecavaptan

Pecavaptan is a vasopressin receptor antagonist.
T61852 hCAIX-IN-8

hCAIX-IN-8 (compound 7i) is a highly potent and selective inhibitor of hCAIX, demonstrating potent inhibitory activity against CAIX with an IC50 value of 0.024 μM. It also exhibits inhibitory activity against CAII and CAVA with IC50 values of 1.99 μM and 1.10 μM, respectively. Furthermore, hCAIX-IN-8 exhibits anti-proliferative effects and low toxicity. It effectively reduces the occurrence of epithelial-to-mesenchymal transitions and promotes apoptosis. Additionally, hCAIX-IN-8 effectively inhi...
T71641 BMS-593214

BMS-593214 是一种活性位点定向因子 (F)VIIa 抑制剂。BMS-593214 具有抗血栓和抗出血特性。BMS-593214 是人 FVIIa 的直接竞争性抑制,也是 VIIa 激活底物 FX 的非竞争性抑制剂。BMS-593214 预防电诱导颈动脉血栓形成 (AT)、线诱导腔静脉血栓形成 (VT)。

化合物

Excavatin M
Cat.No: T125203
Synonym:
Target:
Pecavaptan
Cat.No: T70066
Synonym:
Target:
hCAIX-IN-8
Cat.No: T61852
Synonym:
Target:
BMS-593214
Cat.No: T71641
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
TN5704 Cavaol E

Cavaol E 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN5704,CAS号为 1233044-20-6。

天然产物

Cavaol E
Cat.No: TN5704
Synonym:
Target:
Cat. No. Product Name Species Expression System
TMPY-01877 CA5A Protein, Human, Recombinant (His)

CA5,GS1-21A4.1,CA5AD,carbonic anhydrase VA, mitochondrial,CA...

Human E. coli
Carbonic anhydrase 5A, mitochondrial, also known as Carbonate dehydratase VA, Carbonic anhydrase VA, CA-VA and CA5A, is a member of thealpha-carbonic anhydrase family. Carbonic anhydrases (CAs) are a large family of zinc metalloenzymes first discovered in 1933 that catalyze the reversible hydration of carbon dioxide. CAs participate in a variety of biological processes, including respiration, calcification, acid-base balance, bone resorption, and the formation of aqueous humor, cerebrospi...

重组蛋白

CA5A Protein, Human, Recombinant (His)
Cat.No: TMPY-01877
Species: Human
Expression System: E. coli
TargetMol Loading
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