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抑制剂 & 化合物

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天然产物

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Cat. No. Product Name Target Signaling Pathways
TP1913 BA 1

Potent bombesin receptor agonist (IC50 values are 0.26, 1.55 and 2.52 nM for BB1, BB2 and BB3 respectively). Enhances glucose transport in obese and diabetic primary myocytes. Also stimulates NCI-H1299 lung cancer cell proliferation in vitro.
T34640 Silagaba132

Silagaba 132,Silagaba-132

Silagaba132 is a silicon-containing GABA derivative which treats neuropathic pain without central nervous system related side effects.
T34641 Silagaba161

Silagaba-161,Silagaba 161

Silagaba161 is a silicon-containing GABA derivative which treats neuropathic pain without central nervous system related side effects.
T73531 SABA1

SABA1 具有抗菌活性,比如铜绿假单胞菌和大肠杆菌,其对大肠杆菌的IC50值为 4.0 µM。
T8792 SMBA1

SMBA1 是一种 Bax 激活因子,是一种有效的 Bax 激动剂(Ki :43.3 nM),诱导恶性胶质瘤细胞周期阻滞和凋亡。SMBA1 有增强 Bax 表达的作用,显示出抗肿瘤活性。SMBA1 可用于研究癌症。

化合物

BA 1
Cat.No: TP1913
Synonym:
Target:
Silagaba132
Cat.No: T34640
Synonym: Silagaba 132,Silagaba-132
Target:
Silagaba161
Cat.No: T34641
Synonym: Silagaba-161,Silagaba 161
Target:
SABA1
Cat.No: T73531
Synonym:
Target:
SMBA1
Cat.No: T8792
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T23772 Balanol

Ophiocordin,BA1,Azepinostatin,(-)-Balanol,(3R-trans)-Balanol

Balanol is an ATP-competitive Protein Kinase C and Protein Kinase A inhibitor.

天然产物

Balanol
Cat.No: T23772
Synonym: Ophiocordin,BA1,Azepinostatin,(-)-Balanol,(3R-trans)-Balanol
Target:
TargetMol Loading
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