Cat. No. | Product Name | Target | Signaling Pathways |
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TP2093 |
Apelin-36(human)
Apelin-36 (human) |
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Endogenous APJ receptor agonist (EC50 = 20 nM) that is secreted by adipocytes. Binds with high affinity to human APJ receptors expressed in HEK 293 cells (pIC50= 8.61). Involved in regulation of cardiovascular function, fluid homeostasis and feeding. Bloc | |||
TP2094 |
Apelin-36(rat, mouse)
Apelin-36 (rat, mouse) |
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Endogenous APJ receptor agonist that is secreted by adipocytes. Binds with high affinity to APJ receptors (IC50 = 5.4 nM) and potently inhibits cAMP production in vitro (EC50 = 0.52 nM). Involved in regulation of cardiovascular function, fluid homeostasis | |||
T75783 |
Apelin-36(human) TFA
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Apelin-36(human) TFA 是一种内源性孤儿 G 蛋白偶联受体 APJ 激动剂,EC50为 20 nM。Apelin-36(human) TFA 对 HEK 293 细胞表达的人 APJ 受体有很高的亲和力 (pIC50=8.61)。Apelin-36(human) TFA 与两种主要的生物活性有关:心血管和代谢。Apelin-36(human) TFA 抑制 HIV-1和 HIV-2进入表达 APJ 的 NP2/CD4细胞。 | |||
T75784 |
Apelin-36(rat, mouse) TFA
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Apelin-36(rat, mouse) TFA 是一种内源性孤儿 G 蛋白偶联受体 APJ 激动剂。Apelin-36(rat, mouse) TFA 与 APJ 受体结合,IC50为 5.4 nM,显著抑制 cAMP 的产生,EC50为 0.52 nM。Apelin-36(rat, mouse) TFA 阻断 HIV-1和 HIV-2毒株进入表达 APJ 的 NP-2/CD4 细胞。 |