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Cat. No. | Product Name | Target | Signaling Pathways |
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T39868 |
Anticancer agent 11
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Anticancer agent 11 an effective broad-spectrum anticancer agent, exerts its therapeutic potential by suppressing angiogenesis and facilitating the formation of DNA cross-links. | |||
T38474 |
CL2-MMT-SN38
CL2-MMT-SN38 |
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CL2-MMT-SN38 is a derivative of SN-38, which is a potent anticancer agent and the active metabolite of Irinotecan (CPT-11), a Topoisomerase I inhibitor. | |||
T62278 | Anticancer agent 36 | ||
Anticancer agent 36 (compound 11) 是一种有效的抗微生物剂和抗癌剂,是一种磺酰脲类衍生物。Anticancer agent 36 对蕈状芽孢杆菌、大肠杆菌和白色念珠菌的微生物生长有抑制作用 (MIC: 0.156 - 0.039 mg/mL)。Anticancer agent 36 能够抑制 A549 细胞 (IC50: 19.7 μg/mL)、PC3 细胞 (IC50: 11.9 μg/mL) 生长。 | |||
T78972 |
Anticancer agent 111
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Anticanceragent 111(compound 11)作为一种细胞色素P450抑制剂,对CYP3A4具有3 μM的IC50值,显示出抗癌活性,并可应用于癌症研究。 | |||
T79322 | Antiproliferative agent-30 | ||
Antiproliferative agent-30 (Compound 8g) 抑制微管蛋白组装且可抑制FLT3及Abl1。该化合物展现出对血管的破坏活性,并对多种癌细胞系表现出强效的抗增殖能力,包括HCT-116、K562及MV-4-11细胞(IC50值分别为0.054 nM、0.008 nM、0.144 nM)。此外,Antiproliferative agent-30 亦对携带FLT3-ITD-TKD突变的AML显示出抗癌效果。 |
Cat. No. | Product Name | Target | Signaling Pathways |
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T83088 |
Anticancer agent 156
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Anticanceragent 156(compound 11)是一种基于Miliusanes的强效抗癌剂,有效抑制人源癌细胞生长,并对胃癌细胞展现出显著细胞毒性。 |