Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T13561 | AT6 | Others | Others |
AT6 is a PROTAC AT1 analog which is a highly selective bromodomain (Brd4) degrader. | |||
T79185 |
STAT6-IN-2
|
STAT | JAK/STAT signaling; Stem Cells |
STAT6-IN-2 (Comp R-84) 是STAT6的一种抑制剂,能够抑制嗜酸粒细胞趋化因子-3的分泌,常用于免疫疾病研究。 | |||
T70919 |
NAT6-297775
|
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NAT6-297775 is a SHP2 inhibitor with IC50 =2.47uM. | |||
T73129 |
STAT6-IN-1
|
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STAT6-IN-1(化合物19a)是一种针对STAT6的SH2结构域表现出较高亲和力(IC50=0.028 µM)的STAT6抑制剂。该化合物主要用于研究过敏性肺病、过敏性鼻炎、慢性阻塞性肺病或癌症。 | |||
T15644 |
KAT681
T0681 |
Thyroid hormone receptor(THR) | Endocrinology/Hormones |
KAT681 is a liver selective thyromimetic. | |||
T75146 | KAT6-IN-1 | ||
KAT6-IN-1 是一种有效的KAT6抑制剂。KAT6-IN-1可用于癌症研究。 | |||
T79186 | STAT6-IN-3 | STAT | JAK/STAT signaling; Stem Cells |
STAT6-IN-3 (Compound 18a),一种针对STAT6的Src同源2 (SH2) 结构域的抑制剂,具有44 nM的IC50值。该化合物主要适用于研究哮喘等炎症性疾病。 |