Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T23752 |
AR-C141990
ARC-141990,AR C141990,ARC141990,ARC 141990 |
||
AR-C141990 is a lactate transporters inhibitor. | |||
T37822 | AR-C 141990 hydrochloride | ||
Monocarboxylate transporter (MCT1) inhibitor (pKi = 7.6. Exhibits approximately 10-fold selectivity for MCT1 over MCT2 and no significant activity against MCT3 or 4. Inhibits graft versus host response and prolongs cardiac graft survival in a rat model. Immunosuppressant. Also inhibits brain penetration of GHB analog HOCPCA. |