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Targets Recommended: Aquaporin PROTAC Linker

3

抑制剂 & 化合物

2

重组蛋白

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Cat. No. Product Name Target Signaling Pathways
T5102 TGN-020

TGN020

Aquaporin; PROTAC Linker Membrane transporter/Ion channel; PROTAC
TGN-020 是一种属于 alkyl chain 类的 PROTAC linker,可用于 PROTAC 的合成分子。TGN020 是一种选择性水通道蛋白 4 (AQP4) 抑制剂,IC50为 3.1 μM。TGN020 减轻大鼠脊髓压迫损伤后的水肿并抑制神经胶质瘢痕的形成。
T7946 AER-271

Aquaporin Membrane transporter/Ion channel
AER-271 是一种 AER-270 的膦酸酯前药,是aquaporin-4抑制剂,有用于急性缺血性中风的研究潜力。
T69387 NMO-IgG blocker A-01

NMO-IgG blocker A-01 is a idiotype-specific blocker of neuromyelitis opticaimmunoglobulin g (nmo-igg) binding to aquaporin-4 (aqp4)

化合物

TGN-020
Cat.No: T5102
Synonym: TGN020
Target: Aquaporin, PROTAC Linker
AER-271
Cat.No: T7946
Synonym:
Target: Aquaporin
NMO-IgG blocker A-01
Cat.No: T69387
Synonym:
Target:
Cat. No. Product Name Species Expression System
TMPH-02980 Aquaporin-4/AQP4 Protein, Mouse, Recombinant (His)

Mercurial-insensitive water channel,Aquaporin-4,WCH...

Mouse P. pastoris (Yeast)
Aquaporin-4/AQP4 Protein, Mouse, Recombinant (His) is expressed in yeast with N-6xHis tag. The predicted molecular weight is 9.9 kDa and the accession number is P55088.
TMPH-00953 Aquaporin-4/AQP4 Protein, Human, Recombinant (His & SUMO)

Aquaporin-4,WCH4,AQP-4,M...

Human E. coli
Aquaporin-4/AQP4 Protein, Human, Recombinant (His & SUMO) is expressed in E. coli.

重组蛋白

Aquaporin-4/AQP4 Protein, Mouse, Recombinant (His)
Cat.No: TMPH-02980
Species: Mouse
Expression System: P. pastoris (Yeast)
Aquaporin-4/AQP4 Protein, Human, Recombinant (His & SUMO)
Cat.No: TMPH-00953
Species: Human
Expression System: E. coli
TargetMol Loading
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