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Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T5102 |
TGN-020
TGN020 |
Aquaporin; PROTAC Linker | Membrane transporter/Ion channel; PROTAC |
TGN-020 是一种属于 alkyl chain 类的 PROTAC linker,可用于 PROTAC 的合成分子。TGN020 是一种选择性水通道蛋白 4 (AQP4) 抑制剂,IC50为 3.1 μM。TGN020 减轻大鼠脊髓压迫损伤后的水肿并抑制神经胶质瘢痕的形成。 | |||
T7946 |
AER-271
|
Aquaporin | Membrane transporter/Ion channel |
AER-271 是一种 AER-270 的膦酸酯前药,是aquaporin-4抑制剂,有用于急性缺血性中风的研究潜力。 | |||
T69387 |
NMO-IgG blocker A-01
|
||
NMO-IgG blocker A-01 is a idiotype-specific blocker of neuromyelitis opticaimmunoglobulin g (nmo-igg) binding to aquaporin-4 (aqp4) |
Cat. No. | Product Name | Species | Expression System |
---|---|---|---|
TMPH-02980 |
Aquaporin-4/AQP4 Protein, Mouse, Recombinant (His)
Mercurial-insensitive water channel,Aquaporin-4,WCH... |
Mouse | P. pastoris (Yeast) |
Aquaporin-4/AQP4 Protein, Mouse, Recombinant (His) is expressed in yeast with N-6xHis tag. The predicted molecular weight is 9.9 kDa and the accession number is P55088. | |||
TMPH-00953 |
Aquaporin-4/AQP4 Protein, Human, Recombinant (His & SUMO)
Aquaporin-4,WCH4,AQP-4,M... |
Human | E. coli |
Aquaporin-4/AQP4 Protein, Human, Recombinant (His & SUMO) is expressed in E. coli. |