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Targets Recommended: Antifungal

3

抑制剂 & 化合物

1

重组蛋白

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Cat. No. Product Name Target Signaling Pathways
T61355 APX2039

APX-2039,APX 2039

Antifungal Microbiology/Virology
APX2039 是一种口服有效的真菌 Gwt1 酶 (fungal Gwt1 enzyme) 抑制剂,是新型Gwt2096抑制剂APX1的前药。APX2039 对 C. neoformans 和 C. gattii 展现出极强的抗氪球菌活性。APX2039 具有有效的抗真菌活性,科阻断 GPI (糖基磷脂酰肌醇)锚定细胞壁甘露蛋白的定位。APX2039 可用于研究隐球菌脑膜炎 (CM) 。
T70732 APX2014

APX2014 is a novel potent and specific Ref-1 inhibitor, blocking in vitro cell proliferation and activating apoptosis via PARP cleavage.
T70733 APX2009

APX2009 is a second-generation APE1/Ref-1 redox-specific inhibitor. APX2009 significantly reduces NFkB transcriptional activity, survivin mRNA, and survivin protein levels. APX2009 decreases prostate cancer cell proliferation and induces cell cycle arrest.

化合物

APX2039
Cat.No: T61355
Synonym: APX-2039,APX 2039
Target: Antifungal
APX2014
Cat.No: T70732
Synonym:
Target:
APX2009
Cat.No: T70733
Synonym:
Target:
Cat. No. Product Name Species Expression System
TMPH-00096 APX2, cytosolic Protein, Arabidopsis thaliana, Recombinant (His)

APX1b,APX2,L-ascorbate peroxidase...

Arabidopsis thaliana E. coli
APX2, cytosolic Protein, Arabidopsis thaliana, Recombinant (His) is expressed in E. coli expression system with N-6xHis tag. The predicted molecular weight is 31.5 kDa and the accession number is Q1PER6.

重组蛋白

APX2, cytosolic Protein, Arabidopsis thaliana, Recombinant (His)
Cat.No: TMPH-00096
Species: Arabidopsis thaliana
Expression System: E. coli
TargetMol Loading
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