Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T79504 |
AMPA receptor modulator-6
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iGluR | Membrane transporter/Ion channel; Neuroscience |
AMPA receptormodulator-6 (化合物 (R,R)-2b) 作为一种AMPA受体正向变构调节剂 (AMPA receptor PAM),可应用于神经系统性疾病的研究领域。 | |||
T36809 |
UoS 12258
|
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Positive allosteric modulator of AMPA receptors (pEC50 = 5.2 for potentiation of AMPA-mediated currents in vitro). Also potentiates AMPA-mediated synaptic responses in vivo. Improves performance of rats in various learning and memory paradigms Ward et al (2010) Discovery of N-[(2S)-5-(6-fluoro-3-pyridinyl)-2,3-dihydro-1H-inden-2-yl]-2-propanesulfonamide, a novel clinical AMPA receptor positive modulator. J.Med.Chem. 53 5801 PMID:20614889 |Ward et al (2017) Pharmacological characterization of N-[... |