Cat. No. | Product Name | Target | Signaling Pathways |
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T79191 | AMPA receptor modulator-5 | iGluR | Membrane transporter/Ion channel; Neuroscience |
AMPA receptormodulator-5 (Example 217) 为一种AMPA receptor调节剂,适用于神经系统疾病研究。 | |||
T36809 |
UoS 12258
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Positive allosteric modulator of AMPA receptors (pEC50 = 5.2 for potentiation of AMPA-mediated currents in vitro). Also potentiates AMPA-mediated synaptic responses in vivo. Improves performance of rats in various learning and memory paradigms Ward et al (2010) Discovery of N-[(2S)-5-(6-fluoro-3-pyridinyl)-2,3-dihydro-1H-inden-2-yl]-2-propanesulfonamide, a novel clinical AMPA receptor positive modulator. J.Med.Chem. 53 5801 PMID:20614889 |Ward et al (2017) Pharmacological characterization of N-[... |