Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T6278 |
Sotrastaurin
索曲妥林,AEB071 |
PKC | Chromatin/Epigenetic; Cytoskeletal Signaling |
Sotrastaurin (AEB071) 是一种口服有效的泛 PKC 抑制剂,对 PKCθ、PKCβ、PKCα、PKCη、PKCδ 和 PKCε,Ki 分别为 0.22、0.64、0.95、1.8、2.1 和 3.2 nM。 | |||
T24815 |
Sotrastaurin acetate
|
||
Sotrastaurin acetate is a pan-protein kinase C inhibitor. It also has potential immunosuppressive and antineoplastic activities. |