Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T10240 |
ACP-5862
|
BTK | Angiogenesis; Tyrosine Kinase/Adaptors |
ACP-5862 is a major active and pyrrolidine ring-opened metabolite of Acalabrutinib (IC50: 5.0 nM for BTK). Acalabrutinib is an irreversible and highly selective BTK inhibitor (IC50: 3 nM; EC50: 8 nM). |