Cat. No. | Product Name | Target | Signaling Pathways |
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T26536 |
AC-178335
AC 178335,AC178335 |
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AC-178335 is a pure somatostatin (SRIF) antagonist with an affinity constant (Ki) of 172 +/- 12 nM. AC-178335 blocks SRIF inhibition of adenylate cyclase in vitro (IC50 = 5.1 +/- 1.4 microM). It induces GH release when given alone (50 micrograms intraveno |