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抑制剂 & 化合物

重组蛋白

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Cat. No.	Product Name	Target	Signaling Pathways
T62348	A1AR antagonist 3
	A1AR antagonist 3 (compound 13) 是一种选择性的腺苷酸 1 (A1) 受体拮抗剂，作用于人 A1 (Ki: 9.69 nM) 和大鼠 A1 (Ki: 0.529 nM)。A1AR antagonist 3 能够用于研究神经性疾病。
T60915	A1AR antagonist 5
	A1AR antagonist 5 (化合物 20) 是A1 腺苷受体(A1AR)的有效选择性拮抗剂，其pKi 值为 6.11，pIC50值为 5.83。
T60615	A1AR antagonist 6
	A1AR antagonist 6 (化合物 15) 是 A1 腺苷受体(A1AR)的有效的选择性拮抗剂，其pKi 值为 7.13，pIC50值为 6.38。
T72661	A1AT modulator 2
	A1AT modulator 2, 作为A1AT (α-1 antitrypsin) 的调节剂，具有IC50值大于1.0 μM以及EC50值小于0.4 μM。它主要应用于感染和炎症的研究领域。
T60687	A1AR antagonist 1
	A1AR antagonist 1 (compound 18g) 是A1腺苷受体的选择性拮抗剂。A1AR antagonist 1对 hA1, hA2A，hA2B 受体的Ki 值分别为 2.08、6.91 和 31.2 nM。
T60580	A1AR antagonist 2
	A1AR antagonist 2 (compound 18h) 是 A1腺苷受体 (A1 adenosine receptor) 的有效的选择性拮抗剂。A1AR antagonist 2对于 hA1, hA2A，hA2B 的Ki 值分别为 1.49、10.2 和 50.1 nM。
T83227	A1AT modulator 1
	A1AT modulator 1是一种有效的Z ai-抗胰蛋白酶聚合抑制剂，其pIC50值达到8.3。
T61536	A1AR antagonist 4
	A1AR antagonist 4 (compound 22) is a highly developed chemical compound that acts as a potent and selective antagonist of the A1 adenosine receptor (A1AR). It possesses a pIC50 value of 5.51 and a pKi value of 6.29 [1].
T27509	GW-493838 GW 493838X,GW 493838,GW493838,GW493838X,GW-493838X	Adenosine Receptor	GPCR/G Protein; Neuroscience
	GW-493838是一种有效的腺苷 A1A 受体激动剂，用于治疗血脂异常和神经性疼痛，对创伤或手术引起的疱疹后神经痛或周围神经损伤具有镇痛效果。

化合物

Synonym: GW 493838X,GW 493838,GW493838,GW493838X,GW-493838X

Target: Adenosine Receptor

Species：

Expression System：

Tag：

Cat. No.	Product Name	Species	Expression System
TMPJ-00452	Serpin A1a Protein, Mouse, Recombinant (His) Alpha-1-antitrypsin 1-1, Alpha-1 protease inhibitor 1, Alpha...	Mouse	HEK293 Cells
	Serpin A1a is also known as alpha-1-antitrypsin, is a member of the serpin superfamily of serine proteinase inhibitors that are involved in the regulation of a number of proteolytic processes. Its primary target is elastase, but it also has a moderate affinity for plasmin and thrombin.
TMPY-00915	Serpin A1 Protein, Human, Recombinant (His) PRO2275,SerpinA1,serpin peptidase inhibitor, clade A (alpha-...	Human	HEK293 Cells
	Serpin A1 Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 45.7 kDa and the accession number is P01009-1.
TMPH-00892	A1AR Protein, Human, Recombinant (His) Adenosine receptor A1,ADORA1	Human	E. coli
	Receptor for adenosine. The activity of this receptor is mediated by G proteins which inhibit adenylyl cyclase. A1AR Protein, Human, Recombinant (His) is expressed in E. coli expression system with N-10xHis tag. The predicted molecular weight is 39.3 kDa and the accession number is P30542.