Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T79350 | MAT2A-IN-12 | Methionine Adenosyltransferase (MAT) | Chromatin/Epigenetic |
MAT2A Allosteric inhibitor 2是一种有效的、选择性MAT2A变构抑制剂,具有5 nM的IC50值。在增殖试验(MTAP-/-细胞系)中,MAT2A Allosteric inhibitor 2表现出纳摩尔级别的活性,IC50为5 μM。 |