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抑制剂 & 化合物

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天然产物

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Cat. No. Product Name Target Signaling Pathways
T10663 Calcitriol-d6

Calcitriol D6,骨化三醇 D6

Others Others
Calcitriol D6 is the deuterated form of Calcitriol, which is the hormonally active form of vitamin D. Calcitriol is the active metabolite of vitamin D3 that activates the vitamin D receptor.
T35524 (1S)-Calcitriol

(1S)-Calcitriol (1α,25-Dihydroxy-3-epi-vitamin-D3) is a natural metabolite of 1α,25-dihydroxyvitamin D3 (1α,25(OH)2D3). (1S)-Calcitriol exhibits potent vitamin D receptor (VDR)-mediated actions such as inhibition of keratinocyte growth or suppression of parathyroid hormone secretion[1]. 3‐epi‐Calcitroic acid is an end product of (1S)-Calcitriol (1α,25-Dihydroxy-3-epi-vitamin-D3; 3‐epi‐1a,25(OH)2D3) metabolism by rat CYP24A1[1]. [1]. Steve Y Rhieu, et al. Metabolic stability of 3-epi-1α,25-dihydr...

化合物

Calcitriol-d6
Cat.No: T10663
Synonym: Calcitriol D6,骨化三醇 D6
Target: Others
(1S)-Calcitriol
Cat.No: T35524
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T6316 Calcitriol

Topitriol,Rocaltrol,Calcijex,RO215535,骨化三醇,1,25-Dihydroxyvitamin D3

Endogenous Metabolite Metabolism
Calcitriol (1,25-Dihydroxyvitamin D3) 是一种维他命 D 的代谢物,一种维他命 D 受体 (VDR) 的激动剂 (IC50=0.4 nM)。Calcitriol 增加肠道对钙和磷的吸收,并与甲状旁腺激素一起增加了骨吸收。

天然产物

Calcitriol
Cat.No: T6316
Synonym: Topitriol,Rocaltrol,Calcijex,RO215535,骨化三醇,1,25-Dihydroxyvitamin D3
Target: Endogenous Metabolite
TargetMol Loading
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