Cat. No. | Product Name | Target | Signaling Pathways |
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T39482 |
Casein Kinase inhibitor A86
Casein Kinase inhibitor A86 |
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Casein Kinase inhibitor A86 is a highly effective and orally bioavailable inhibitor of casein kinase 1α (CK1α). Additionally, it displays inhibitory actions towards CDK7 (TFIIH) and CDK9 (P-TEFb). Furthermore, Casein Kinase inhibitor A86 demonstrates the ability to induce apoptosis in leukemia cells, portraying substantial anti-leukemic effects. |