Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
TNU0327 |
2-Trifluoromethyl adenosine
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Nucleoside Derivatives –8-substituted purine nucleosides ;ara-nucleosides. | |||
T9330 |
MIPS521
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Adenosine Receptor | GPCR/G Protein; Neuroscience |
MIPS521 ({2-Amino-4-[3,5-bis(trifluoromethyl)phenyl]thiophen-3-yl}(4-chlorophenyl)methanone) 是腺苷受体 (A1AR) 的正向变构调节剂,通过调节大鼠脊髓中内源性腺苷水平的升高,在体内表现出减轻疼痛的作用。 | |||
TNU0515 |
2’-Chloro-N6-(4-trifluoromethyl)benzyl adenosine
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2'-Chloro-N6-(4-trifluoromethyl)benzyl adenosine is a Nucleoside Derivative - Halo-nucleoside;2-Modified purine nucleoside; 6-Modified purine nucleoside;. | |||
T75035 | 2’-Chloro-N6-(3-trifluoromethyl)benzyl adenosine | ||
2’-Chloro-N6-(3-trifluoromethyl)benzyl adenosine是一种嘌呤核苷类似物,以其广泛的抗肿瘤活性而知名,特别是针对惰性淋巴系统的恶性肿瘤。其作用机制主要通过抑制DNA合成、诱导细胞凋亡(apoptosis)等方式发挥。 | |||
TNU0514 |
2’-Chloro-N6-(3-trifluoromethyl)benzyl adenosine
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2'-Chloro-N6-(3-trifluoromethyl)benzyl adenosine is a Nucleoside Derivative - Halo-nucleoside;2-Modified purine nucleoside; 6-Modified purine nucleoside;. |