Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T7215 |
NM107
NM-107,2'-C-甲基胞嘧啶核苷,2'-C-Methylcytidine |
HCV Protease | Microbiology/Virology; Proteases/Proteasome |
NM107 (2'-C-Methylcytidine) 是一种具有广谱抗病毒活性的核糖核苷,是丙型肝炎病毒 NS5B 聚合酶的核苷抑制剂,在野生型复制子细胞中的 EC50 为 1.85 μM。 | |||
T38237 |
2′-O-Methylcytidine
|
Nucleoside Antimetabolite/Analog; HCV Protease | Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology; Proteases/Proteasome |
2'-O-Methylcytidine 是 2'-代核苷,可抑制 HCV 复制。 它在体外抑制 NS5B 催化的 RNA 合成,其抑制方式是与底物核苷三磷酸竞争。 | |||
TNU0308 | N4-Amino-2’-C-methylcytidine | ||
Nucleoside Derivatives - 2’-Modified nucleosides; Amino-nucleosides | |||
T13281 |
Valopicitabine
NM283 |
HCV Protease | Microbiology/Virology; Proteases/Proteasome |
Valopicitabine is an effective prodrug of the effective anti-HCV drug 2'-C-methylcytidine and can be used as a promising antiviral drug for the study of chronic HCV infection. |