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Cat. No. Product Name Target Signaling Pathways
T70267 ADL 08-0011 HCl

ADL 08-0011 is an active metabolite of the μ-opioid receptor antagonist alvimopan. It is produced from alvimopan via amide hydrolysis by gut microbiota. ADL 08-0011 is a μ-opioid receptor antagonist (Ki = 0.25 nM). It is selective for μ-opioid receptors over κ- and δ-opioid receptors (Kis = 15.8 and 31.6 nM, respectively). ADL 08-0011 inhibits endomorphin 1-induced inhibition of electrically induced contraction of isolated guinea pig ileum (pA2 = 9.4). In vivo, ADL 08-0011 (0.03-1 mg/kg) reverse...
T20081 ADL-08-0011

ADL 08-0011

ADL-08-0011 is an metabolite of alvimopan.

化合物

ADL 08-0011 HCl
Cat.No: T70267
Synonym:
Target:
ADL-08-0011
Cat.No: T20081
Synonym: ADL 08-0011
Target:
TargetMol Loading
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