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Cat. No. Product Name Target Signaling Pathways
T38841 IRE1α kinase-IN-2

IRE1α kinase-IN-2

IRE1α kinase-IN-2 is a highly potent inhibitor of IRE1α kinase, demonstrating an EC50 of 0.82 μM. It effectively impedes IRE1α kinase autophosphorylation with an IC50 of 3.12 μM. Additionally, IRE1α kinase-IN-2 effectively inhibits the splicing of XBP1 mRNA in wild-type cell lines.

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IRE1α kinase-IN-2
Cat.No: T38841
Synonym: IRE1α kinase-IN-2
Target:
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