Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T10320 |
Androgen receptor antagonist 1
|
Others | Others |
Androgen receptor antagonist 1 is an orally available full androgen receptor antagonist (IC50: 59 nM). It can be used in the synthesis of PROTAC AR degraders, which results in 24% and 47 % AR protein degradation in LNCaP cells at 1 μM and 10 μM, respectively. |