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Cat. No. Product Name Target Signaling Pathways
T64234 Alosetron (Hydrochloride(1:X))

Alosetron (GR 68755) Hydrochloride (1:X) 是一种高效的、具有高度选择性的、具有抗炎作用的 5-HT3 受体 (5-HT3 receptor) 拮抗剂。Alosetron Hydrochloride (1:X) 能够阻断 5HT3 介导的豚鼠肌间和粘膜下神经元的快速去极化(IC50:~55 nM)。Alosetron Hydrochloride (1:X) 能够减缓清醒或麻醉犬直肠扩张的内脏伤害性效应。Alosetron Hydrochloride (1:X) 能够用于研究肠易激综合征 (IBS)。
T21235 Alosetron

Lotronex,GR68755,GR-68755,GR 68755,阿洛司琼

Alosetron, a 5-HT3 antagonist, is used for the management of severe diarrhea-predominant irritable bowel syndrome (IBS) in women only.
T19190 Alosetron D3 Hydrochloride

GR-68755C D3

Others Others
Alosetron D3 (GR 68755 D3) Hydrochloride is a deuterium-labeled Alosetron. Alosetron is an antagonist of 5HT3-receptor.
T19191 Alosetron-d3

Alosetron D3,GR 68755 D3,GR 68755X D3

Others Others
Alosetron D3 (GR 68755 D3) is a deuterium-labeled Alosetron. Alosetron is an antagonist of 5HT3-receptor.

化合物

Alosetron (Hydrochloride(1:X))
Cat.No: T64234
Synonym:
Target:
Alosetron
Cat.No: T21235
Synonym: Lotronex,GR68755,GR-68755,GR 68755,阿洛司琼
Target:
Alosetron D3 Hydrochloride
Cat.No: T19190
Synonym: GR-68755C D3
Target: Others
Alosetron-d3
Cat.No: T19191
Synonym: Alosetron D3,GR 68755 D3,GR 68755X D3
Target: Others
TargetMol Loading
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