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抑制剂 & 化合物

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天然产物

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Cat. No. Product Name Target Signaling Pathways
T37433 Erythromycin lactobionate

Erythromycin is a macrolide antibiotic that inhibits bacterial protein synthesis by targeting the 50S ribosomal subunit, blocking the progression of nascent polypeptide chains.[1] It is effective against a host of bacterial genera, including Streptococcus, Staphylococcus, and Haemophilus (MIC90s range from 0.015-2.0 mg/l).[2] Erythromycin is known to potently inhibit the cytochrome P450 isoform CYP3A4, which can affect the metabolism of numerous clinically relevant medications.[3],[4] Erythromyc...
T69688 Erythromycin Gluceptate

Erythromycin Gluceptate is an inhibitor of protein translation and mammalian mRNA splicing. It inhibits growth of gram negative and gram positiove bacteria.
T70696 Erythromycin hydrochloride

Erythromycin hydrochloride is an inhibitor of protein translation and mammalian mRNA splicing. It inhibits growth of gram negative and gram positiove bacteria.

化合物

Erythromycin lactobionate
Cat.No: T37433
Synonym:
Target:
Erythromycin Gluceptate
Cat.No: T69688
Synonym:
Target:
Erythromycin hydrochloride
Cat.No: T70696
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T1032 Erythromycin

红霉素,E-Mycin

ribosome; Antibacterial; Antibiotic Microbiology/Virology
Erythromycin (E-Mycin) 是由放线菌产生的大环内酯类抗生素。它结合细菌的 50S 核糖体亚基,通过阻断转肽和易位反应来抑制 RNA 依赖性蛋白的合成。
T15245 Erythromycin estolate

Phtalic anhydride,ilosone

Antibacterial Microbiology/Virology
Erythromycin estolate 是红霉素的衍生物,属于大环内酯类抗生素,常用于研究多种细菌感染。酯酸红霉素对胆汁酸转运有抑制作用,可引起肝损伤,主要是胆汁淤积性肝炎。

天然产物

Erythromycin
Cat.No: T1032
Synonym: 红霉素,E-Mycin
Target: ribosome, Antibacterial, Antibiotic
Erythromycin estolate
Cat.No: T15245
Synonym: Phtalic anhydride,ilosone
Target: Antibacterial
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