Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T22433 |
Sulopenem
CP-70429,硫培南 |
Others | Others |
Sulopenem, an orally active, potent inhibitor of beta-lactamase, is a parenteral penem antibiotic with broad-spectrum activities against Gram-negative and Gram-positive bacteria. | |||
T78987 |
SA09-Cu
|
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SA09-Cu是一种NDM-1的非竞争性抑制剂,具有9.6 nM的IC50。该化合物通过作用于氧化酶的Zn(II)-硫醇盐位点,能将NDM-1转化为无活性形态,从而抵御细菌细胞内的硫醇还原作用。SA09-Cu对于多种产生NDM-1的肠杆菌科碳青霉烯耐药菌株(CRE)表现出明显的抑制作用,有效恢复了美罗培南的活性,并有助于减缓碳青霉烯耐药性的进展。 |